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  Annoucement
 
24 May, 2010
KAMETANI AWARD 2010
Presented to Prof. Kozo Shishido

For Outstanding Research In Heterocyclic Chemistry
And Contributions to the Heterocycles.

The Nomination commitiee of Heterocycles is pleased to announce that for 2010, the Kametani Award has been awarded to Prof. Kozo Shishido for his outstanding research in Heterocyclic Chemistry and contributions to Heterocycles.

The Kametani Award was founded in 1999 by the Memory of the founder of Heterocycles.
Sponsored by The Japan Institute of Heterocyclic Chemistry and Elsevier

 
 
30 November, 2009
The 6th Eurasian Meeting on Heterocyclic Chemistry (6th EAMHC) will be held at Alicante (Spain)

June 30-July 4, 2010.

The aim of this meeting is to cover a wide range of topics of current interest in the field of heterocyclic chemistry.
Chairman: Prof. Dr.Miguel Yus,
Co-Chairman: Prof. Dr. Carmen Nájera
More information:

http://web.ua.es/en/ 6theamhc/presentation.html

 
 
 
  Archive
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 Prepress The most recently 20 articles Free PDF 
 
29 July, 2010 (Vol. 82, Special issue)
Paper
Preparation of Highly Conjugated Oligoaza-PAHs Based on the Oxidative Intramolecular Coupling of Bicyclo[2.2.2]octadiene-Fused Pyrrole
Hidemitsu Uno,* Takahiro Takiue, Hiroki Uoyama, Tetsuo Okujima, Hiroko Yamada, and Go Masuda
DOI: 10.3987/COM-10-S(E)69
Abstract     Supporting Info. (271KB)    PDF (1MB)
 

Paper
A Facile Synthesis of Fluorine-Containing 1,7-Phenanthrolines by the Cyclization of N-Propargyl-6,8-bis(trifluoroacetyl)quinolin-5-amine with Various Active Methylene Compounds
Dai Shibata, Ayaka Sakai, Mizuki Hatakenaka, Shohei Saikawa, Yasuhiro Kamitori, Maurice Médebielle, and Etsuji Okada*
DOI: 10.3987/COM-10-S(E)71
Abstract     PDF (651KB)
 

Note
Convenient Synthesis of Optically Pure 8-Methoxy-2-methyl-1,2,3,4-tetrahydroquinoline and 2-Methyl-1,2,3,4-tetrahydroquinoline
Jie Tang, Guo-Fang Jiang,* and Yong-Gui Zhou*
DOI: 10.3987/COM-10-S(E)50
Abstract     PDF (614KB)
 

Communication
Enantioselective Synthesis of the C(2)-C(11) Cyclopropylfuran Segment of Pinnatin A
Masayoshi Tsubuki,* Terunobu Abekura, Kazunori Takahashi, and Toshio Honda*
DOI: 10.3987/COM-10-S(E)91
Abstract     PDF (2.4MB)
 

27 July, 2010 (Vol. 82, Special issue)
Communication
Synthesis of 2,3,4-Tri-Substituted 3,4-Dihydroquinazolines via Tandem Nucleophilic Addition/Epoxy Ring-Opening Cyclization Methodology Using N-(2-Oxiranylphenyl)carbodiimides with Nucleophiles
Takao Saito,* Tatsuya Ote, Masahiro Shiotani, Hiroko Kataoka, Takashi Otani, and Noriki Kutsumura
DOI: 10.3987/COM-10-S(E)66
Abstract     PDF (282KB)
 

Paper
Stereoselective Synthesis of Caribbean Ciguatoxin M-Ring Using [2+2] Photocyclization
Shuji Yamashita,* Naoya Iijima, Takahiro Shida, and Masahiro Hirama*
DOI: 10.3987/COM-10-S(E)61
Abstract     PDF (1.7MB)
 

Communication
Decarboxylative C-C Bond Cleavage Reactions via Oxapalladacycles
Masanari Kimura,* Tomohiko Kohno, Kei Toyoda, and Takamichi Mori
DOI: 10.3987/COM-10-S(E)46
Abstract     PDF (343KB)
 

Communication
A Novel Synthesis of a 1,3-Disubstituted 1,3-Dihydro-2H-imidazo[4,5-b]pyridin-2-one. Application to GW808990 a CRF1 Receptor Antagonist
Jerome F. Hayes* and Matthew E. Popkin
DOI: 10.3987/COM-10-S(E)62
Abstract     PDF (573KB)
 

22 July, 2010 (Vol. 82, Special issue)
Note
Simple Deuterium Introduction at α-Position of Carbonyl in Diazirinyl Derivatives for Photoaffinity Labeling
Yuta Murai, Miho Takahashi, Yasuyuki Muto, Yasumaru Hatanaka, and Makoto Hashimoto*
DOI: 10.3987/COM-10-S(E)57
Abstract     PDF (261KB)
 

Paper
Crystal-State Structure Analysis of β-Hydroxy-γ-Lactam Constrained Ser/Thr Peptidomimetics
Daniel J. St-Cyr, Thierry Maris, and William D. Lubell*
DOI: 10.3987/COM-10-S(E)52
Abstract     PDF (12.9MB)
 

Communication
An Enantioselective Synthesis of the Resorcyclic Acid Lactone L-783,277 via Addition of an Acetylide Anion to a Tethered Weinreb Amide
Andrew Lin, Anthony C. Willis, and Martin G. Banwell*
DOI: 10.3987/COM-10-S(E)67
Abstract     PDF (347KB)
 

21 July, 2010 (Vol. 82, Special issue)
Paper
Diastereoselective Cyclization Reactions of Chiral Proline Auxiliary-Substituted N-Benzoyl-α-dehydro(1-naphthyl)alaninamide Derivatives via Photoinduced Electron Transfer
Yuhki Sato, Yuhta Haruyama, Tetsutaro Igarashi, and Tadamitsu Sakurai*
DOI: 10.3987/COM-10-S(E)33
Abstract     PDF (430KB)
 

21 July, 2010 (Regular issue)
Note
One-Step Construction of 6-Aza-2-thiabicyclo[3.3.1]nona-3,7-diene Framework
Nagatoshi Nishiwaki* and Kazuya Kobiro
DOI: 10.3987/COM-10-11998
Abstract     PDF (400KB)
 

16 July, 2010 (Vol. 82, Special issue)
Paper
Synthesis of 8,1’-etheno and 8,2’-ethano Bridged Guanosine Derivatives Using Radical Cyclization
Julian Strohmeier, André Nadler, Daniel Heinrich, Ansgar Fitzner, and Ulf Diederichsen*
DOI: 10.3987/COM-10-S(E)51
Abstract     PDF (664KB)
 

Paper
Screening the Structural Space of Bicyclo-DNA: Synthesis and Properties of Bicyclo-DNA Functionalized at C(6’)
Samuel Luisier and Christian J. Leumann*
DOI: 10.3987/COM-10-S(E)65
Abstract     PDF (2.5MB)
 

15 July, 2010 (Regular issue)
Paper
A Novel Pentose Synthesis via Palladium(II)-Catalyzed Cyclization of an Unstable Hemiacetal
Ken-ichiro Awasaguchi, Masahiro Miyazawa,* Ikuyo Uoya, Koichi Inoue, Koji Nakamura, Hajime Yokoyama, and Yoshiro Hirai*
DOI: 10.3987/COM-10-12001
Abstract     PDF (562KB)
 

13 July, 2010 (Vol. 82, Special issue)
Paper
Nucleotides Part: LXXVII New Types of Fluorescence Labeling of 2’-Deoxyguanosine
Thomas Maier and Wolfgang Pfleiderer*
DOI: 10.3987/COM-10-S(E)54
Abstract     PDF (702KB)
 

Note
[2+2+2]-Cocyclotrimerization of 6-Alkynyl-7-benzylpurines with α,ω-Diynes
Stanislav Opekar, Pavel Turek, Radek Pohl, Blanka Klepetářová, Ivan Votruba, Michal Hocek,* and Martin Kotora*
DOI: 10.3987/COM-10-S(E)56
Abstract     Supporting Info. (2.1MB)    PDF (2.5MB)
 

9 July, 2010 (Vol. 82, Special issue)
Communication
Boromycin Derivatives: Synthesis and Antimalarial Activity in vitro and in vivo
Ayumi Tsutsui, Yujiro Furuya, Tomoyasu Hirose, Riyon Kim, Rokurou Masuma, Atsuko Matsumoto, Yoko Takahashi, Aki Ishiyama, Miyuki Namatame, Kazuhiko Otoguro, Satoshi Ōmura,* and Toshiaki Sunazuka*
DOI: 10.3987/COM-10-S(E)55
Abstract     PDF (714KB)
 

9 July, 2010 (Regular issue)
Paper
Cyclization Reactions of 2-Isothiocyanatophenyl Ketones Giving 4-Hydroxyquinoline-2(1H)-thiones and 4-Alkylidene-1,4-dihydro-3,1-benzoxazine-2-thiones
Kazuhiro Kobayashi,* Toshihide Komatsu, Shuhei Fukamachi, and Hisatoshi Konishi
DOI: 10.3987/COM-10-11991
Abstract     PDF (198KB)
 

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