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HETEROCYCLES Special Issue Vol. 105 in honor of Professor Somsak Ruchirawat on 80th Birthday
HETEROCYCLES Special Issue Vol. 105 in honor of Professor Somsak Ruchirawat on 80th Birthday
Submission deadline: December 20, 2021
On the occasion of Professor Somsak Ruchirawat's 80th birthday, HETEROCYCLES editorial office is planning to publish special anniversary issue on June 28, 2022 as Vol. 105. Authors are invited to submit their work to this topical issue.
Authors wishing to submit their manuscript should contact editorial office via e-mail by April 26, 2021. Manuscript should reach the editorial office no later than December 20, 2021.
Contact: submit@heterocycles.com
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e-Journal
Abstract
1 data found. 1 - 1 listed
Paper | Special issue | Vol 86, No. 2, 2012, pp. 1483 - 1494
Published online: 22nd November, 2012
Full Text HTMLPDF (794KB)PDF with Links (1MB)
Published online: 22nd November, 2012
DOI: 10.3987/COM-12-S(N)129
■ ASYMMETRIC INTRAMOLECULAR CONJUGATE ADDITION OF α-AMINO ACID DERIVATIVES VIA RACEMIZATION-FREE EQUILIBRIUM OF INTERMEDIARY CHIRAL ENOLATES
Daiki Monguchi, Tomoyuki Yoshimura, Kazuyuki Irie, Kazuhiro Hayashi, Swapan Majumdar, Takahiro Sasamori, Norihiro Tokitoh, and Takeo Kawabata*
*Institute for Chemical Research, Kyoto University, Uji, Kyoto 611-0011, Japan
Abstract
A highly enantioselective route to a multi-substituted indoline derivative via intramolecular conjugate addition of an α-amino acid derivative has been developed. Enantioselectivity of the reaction was almost independent from the temperature, while the diastereoselectivity was totally dependent on the temperature. High diastereomeric ratios observed at the higher temperatures were assumed to be the results from an equilibrium process between axially chiral enolate intermediates.
1 data found. 1 - 1 listed
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