HETEROCYCLES
An International Journal for Reviews and Communications in Heterocyclic ChemistryWeb Edition ISSN: 1881-0942
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Obituary
Yoshito Kishi (1937-2023)
Yoshito Kishi (1937-2023)
Professor. Yoshito Kishi,
a member of the Honorary Editorial Associates of HETEROCYCLES,
has passed away on January 9, 2023 at the age of 85.
I deeply express my regret over his death.
Kunio Ogasawara
Editor
January 13, 2023
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December 24, 2019
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e-Journal
Abstract
1 data found. 1 - 1 listed
Short Paper | Regular issue | Vol 92, No. 5, 2016, pp. 925 - 935
Published online: 15th March, 2016
PDF (641KB)PDF with Links (845KB)
Published online: 15th March, 2016
DOI: 10.3987/COM-16-13418
■ Novel Twin-Drug Type C2-Symmetrical Phenylboronic Acid Pinacol Esters
Makoto Furutachi, Ayumi Ejima, Reika Tsuru, Saho Goto, Toshiaki Gondo, Kenta Ako, Saya Fujii, Arisa Okumura, Ayumi Tozuka, Kazumi Yokomizo, Jian-Rong Zhou, Hiroshi Inao, Yutaro Ono, Nobuhiro Kashige, Fumio Miake, and Kunihiro Sumoto*
*Faculty of Pharmaceutical Sciences, Fukuoka University, 8-19-1 Nanakuma, Jonan-ku, Fukuoka 814-0180, Japan
Abstract
We here report the preparation of newly designed bivalent twin-drug type C2-symmetrical cyclic phenylboronic acid derivatives. The synthesis of these C2-symmetrical mid-size molecules 3 was accomplished by an amide bond formation reaction using amino-substituted phenylboronic acid pinacol esters 1 and dicarboxylic acid dichlorides 2 in the presence of Et3N. We confirmed that this procedure is conventionally applicable to the preparation of various C2-symmetrical cyclic boronic acid derivatives 3 in good to excellent yields.
1 data found. 1 - 1 listed
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