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■ Synthesis of Quinolyl- and Isoquinolyl Heteroarylamines Using Palladium Catalyzed Suzuki Cross-Coupling Reaction

Ihl Young Choi Lee,* Myung Hee Jung, Hee-Jeong Lim, and Hyo Won Lee*

*Medicinal Chemistry, Korea Research Institute of Chemical Technology, 100 Jang-dong, Yuseong, Daejon 305-600, Korea

Abstract

Quinolyl- and isoquinolylboronic acids are prepared from 5-bromoquinoline and 5-bromoisoquinoline, respectively, via halogen-metal exchange. Suzuki cross-coupling of these compounds with haloheteroarylamine leading to the corresponding heteroarylamine derivatives is described.