HETEROCYCLES
An International Journal for Reviews and Communications in Heterocyclic ChemistryWeb Edition ISSN: 1881-0942
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Paper | Special issue | Vol 70, No. 1, 2006, pp.509-517
Published online, 24th November, 2006■ Synthesis of a Stable Pyridyl Boronate and Its Reaction with Aryl and Heteroaryl Halides
Published online, 24th November, 2006
DOI: 10.3987/COM-06-S(W)54
■ Synthesis of a Stable Pyridyl Boronate and Its Reaction with Aryl and Heteroaryl Halides
Steven J. Durrant,* Joanne L. Pinder,* Jean-Damien Charrier, Juan-Miguel Jimenez, Guy Brenchley, Philip N. Collier, David Kay, Andrew Miller, Françoise Pierard, Sharn Ramaya, Shazia Sadiq, and Heather C. Twin
*Vertex Pharmaceuticals Limited, 88 Milton Park, Abingdon, Oxfordshire, OX14 4RY, U.K.
Abstract
The synthesis and reaction of a versatile 5-pyridyl boronate is described. This intermediate can be used to synthesize a range of biologically interesting 2-(1H)-pyridones.
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