Online article for Non-subscribers

Pay per view

Heterocycles has a pay-per-view service for Non-subscribers.
You will be able to directly purchase the full text article through PayPal.
Your purchased Paper can be downloaded after the payment is completed.
An e-mail will be sent the URL to download the paper.
If you have any questions, please contact: purchase@heterocycles.com

Price: ¥ 4,320 (Yen only)
Period: This Article can be accessed for 7 days.

Paper | Regular issue | Vol 34, No. 7, 1992, pp.1395-1398
Published online, 1st January, 1970
DOI: 10.3987/COM-92-6033
Synthesis of 5-Arylated Indoles via Palladium-catalyzed Cross-coupling Reaction of 5-Indolylboronic Acid with Aryl and Heteroaryl Halides

Youhua Yang and Arnold R. Martin*

*Department of Pharmaceutical Sciences, College of Pharmacy, University of Arizona, Tucson, AZ 85721, U.S.A.

Abstract

Palladium(0)-catalyzed cross-coupling reaction of 5-indolylboronic acid with various aryl and heteroaryl halides results in regioselective formation of 5-arylated indoles in good yields.