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Paper | Regular issue | Vol 34, No. 7, 1992, pp.1395-1398
Published online, 1st January, 1970
DOI: 10.3987/COM-92-6033
Synthesis of 5-Arylated Indoles via Palladium-catalyzed Cross-coupling Reaction of 5-Indolylboronic Acid with Aryl and Heteroaryl Halides

Youhua Yang and Arnold R. Martin*

*Department of Pharmaceutical Sciences, College of Pharmacy, University of Arizona, Tucson, AZ 85721, U.S.A.


Palladium(0)-catalyzed cross-coupling reaction of 5-indolylboronic acid with various aryl and heteroaryl halides results in regioselective formation of 5-arylated indoles in good yields.