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Note | Regular issue | Vol 48, No. 1, 1998, pp.171-174
Published online, 1st January, 1970
DOI: 10.3987/COM-97-7999
One-Pot Access to 2,3-Disubstituted 1,2,3,4-Tetrahydroquinolines by Reductive Amination of Aldehydes with Sodium Cyanoborohydride

Guy Lewin* and Corinne Schaeffer

*Laboratoire de Pharmacognosie, Faculte de Pharmacie, boulevard Becquerel, 14032 Caen, France

Abstract

Slight modification of the reductive amination Borch method (delayed addition of NaBH3CN) provided an easy one-pot synthesis of 1,2,3,4-tetrahydroquinoline derivatives from enolizable aldehydes.