Online article for Non-subscribers

Pay per view

Heterocycles has a pay-per-view service for Non-subscribers.
You will be able to directly purchase the full text article through PayPal.
Your purchased Paper can be downloaded after the payment is completed.
An e-mail will be sent the URL to download the paper.
If you have any questions, please contact: purchase@heterocycles.com

Price: ¥ 4,320 (Yen only)
Period: This Article can be accessed for 7 days.

Paper | Regular issue | Vol 48, No. 9, 1998, pp.1793-1799
Published online, 1st January, 1970
DOI: 10.3987/COM-98-8205
Synthesis of 2-Substituted 3-Alkenyl-indoles by the Palladium-catalyzed Cyclization Followed by Alkenylation (Heck Reaction)

Akito Yasuhara,* Masashi Kaneko, and Takao Sakamoto*

*Faculty of Pharmaceutical Sciences, Tohoku University, Aramaki, Aoba-ku, sendai 980-8578, Japan

Abstract

The reaction of N-protected 2-alkynylanilines with electron-deficient alkenes in the presence of a palladium (II) catalyst and copper dichloride in acetonitrile gave 2-substituted 3-alkenylindoles.