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Obituary
Yoshito Kishi (1937-2023)
Yoshito Kishi (1937-2023)
Professor. Yoshito Kishi,
a member of the Honorary Editorial Associates of HETEROCYCLES,
has passed away on January 9, 2023 at the age of 85.
I deeply express my regret over his death.
Kunio Ogasawara
Editor
January 13, 2023
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Communication | Regular issue | Vol 2, No. 5, 1974, pp.559-563
Published online, 1st January, 1970■ A Novel Formation of 1-Hydroxymethyl-4,5-dimethoxy-7H-azirino[1,2-a]indole-7a-carboxylic Acid γ-Lactone
Published online, 1st January, 1970
DOI: 10.3987/R-1974-05-0559
■ A Novel Formation of 1-Hydroxymethyl-4,5-dimethoxy-7H-azirino[1,2-a]indole-7a-carboxylic Acid γ-Lactone
Tetsuji Kametani,* Frank F. Ebetino, Keiichiro Fukumoto, and Albert I. Meyers
*Pharmaceutical Institute, Tohoku University, Aobayama, Sendai 980-8578, Japan
Abstract
α-(6-Nitroveratrylidene)-γ-butyrolactone (1) rearranges to 3-(6-nitroveratryl)-2(5H)-furanone (5), and is deoxygenated to 1-hydroxymethyl-4,5-dimethoxy-7H-azirino[1,2-a]indole-7a-carboxylic acid γ-lactone (6) in triethyl phosphite at 140 - 150 °. Although frequently postulated in triethyl phosphite reductions of nitro compounds, aziridines have not, heretofore, been isolated.
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