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Paper | Special issue | Vol 90, No. 2, 2015, pp.1038-1071
Published online, 3rd September, 2014
DOI: 10.3987/COM-14-S(K)74
Simple Synthetic Method for 1-Hydroxyindole and Its Application to 1-Hydroxytryptophan Derivatives

Toshiya Kawasaki, Mutsuko Tabata, Kyoko Nakagawa, Kensuke Kobayashi, Atsushi Kodama, Tetsuya Kobayashi, Masakazu Hasegawa, Keiko Tanii, and Masanori Somei*

*Noto Marine Laboratory, Institute of Nature and Environmental Technology, Faculty of Pharmaceutical Sciences, Graduate School of Natural Science and Technology, Kanazawa University, 56-7 Matsuhidai, Matsudo-shi, Chiba 270-2214, Japan


Simple and general synthetic method for 1-hydroxy- and 1-methoxyindole is reported. Its application to the synthesis of various types of 1-hydroxy- and 1-methoxyindole derivatives is successful, especially for the synthesis of 1-hydroxytryptophan derivatives.