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Obituary
Yoshito Kishi (1937-2023)
Yoshito Kishi (1937-2023)
Professor. Yoshito Kishi,
a member of the Honorary Editorial Associates of HETEROCYCLES,
has passed away on January 9, 2023 at the age of 85.
I deeply express my regret over his death.
Kunio Ogasawara
Editor
January 13, 2023
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Paper | Regular issue | Vol 94, No. 6, 2017, pp.1074-1097
Published online, 22nd May, 2017
Published online, 22nd May, 2017
DOI: 10.3987/COM-17-13714
■ Synthesis and Biological Evaluation of Novel Di- and Trisubstituted Thiazole Derivatives
Irmantas Parašotas, Eglė Urbonavičiūtė, Kazimieras Anusevičius, Ingrida Tumosienė, Ilona Jonuškienė, Kristina Kantminienė,* Rita Vaickelionienė, and Vytautas Mickevičius
*Department of Physical and Inorganic Chemistry, Kaunas University of Technology, Radvilenu rd. 19, LT-50254 Kaunas, Lithuania
Abstract
Novel di- and trisubstituted thiazole derivatives bearing heterocyclic, aromatic, chalcone, and carboxyalkyl-heterocyclic moieties were synthesized. Compounds possessing significant antibacterial activity, comparable to that of commercial antibacterial agent ampicillin, against Rhizobium radiobacter, Xanthomonas campestris, and Escherichia coli were identified. Some of the synthesized compounds exhibited a very high antioxidant activity.
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